Zita rechiratidzo | ActiTide™ AH3 |
CAS Nha. | 616204-22-9 |
INCI Zita | Acetyl Hexapeptide-8 |
Application | Lotion, Serums, Mask, Facial cleanser |
Package | 100g / bhodhoro, 1kg / bhegi |
Chitarisiko | Hupfu hwakachena kusvika kuchena |
Solubility | Mvura inonyungudika |
Function | Peptide series |
Sherufu hupenyu | 2 years |
Storage | Chengetedza mudziyo wakavharwa zvakasimba munzvimbo inotonhorera, yakaoma pa2 - 8°C. |
Dosage | 0.005-0.05% |
Application
Tsvagiridzo mumaitiro akakosha ekurwisa kuunyana kwakatungamira mukuwonekwa kweActiTide™ AH3, hexapeptide yekuvandudza yakagadziridzwa kuburikidza nemaitiro esainzi kubva pakugadzira kwakadzikama kusvika pakugadzirwa kweGMP, ine mhedzisiro yakanaka.
ActiTide ™ AH3 inopa kukwenya-kuderedza kushanda kwakafanana neBotulinum Toxin Type A, uku ichidzivirira njodzi dzejekiseni uye ichipa zvakanyanya mutengo-kubudirira.
Cosmetic Benefits:
ActiTide ™ AH3 inoderedza kudzika kwekukwinya kunokonzerwa nekudzvanya kwemhasuru yechiso, iine mhedzisiro pahuma uye periocular wrinkles.
Mechanism of Action:
Tsandanyama contraction inoitika neurotransmitter inoburitswa kubva kune synaptic vesicles. Iyo SNARE yakaoma - musangano weternary weVAMP, Syntaxin, uye SNAP-25 mapuroteni - yakakosha kune vesicle docking uye neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). Iyi yakaoma inoita seya cellular hook, inobata vesicles uye kutyaira membrane fusion.
Sechimiro chemimetic cheSNAP-25 N-terminus, ActiTide™ AH3 inokwikwidza neSNAP-25 kuti ibatanidzwe muSNARE yakaoma, ichigadzirisa gungano rayo. Destabilization yeSNARE yakaoma inokanganisa vesicle docking uye inozotevera neurotransmitter kuburitswa, zvichitungamira kuderedzwa kwemhasuru kudhonzwa uye kudzivirira kwekuwonyana uye mutsara kuumbwa.
ActiTide™ AH3 inzira yakachengetedzeka, ine mari yakawanda, uye yakapfava kune Botulinum Toxin Type A. Inonangana nepamusoro penzira imwechete yekuwunyana asi inoshanda nemuchina wakasiyana.